1: (diethylamino)sulfur trifluoride / CH2Cl2 / 1 h / -78 °C 2: KOH / methanol View Scheme
参考文献
Cravatt, Benjamin F.; Ashley, Jon A.; Janda, Kim D.; Boger, Dale L.; Lerner, Richard A.
Journal of the American Chemical Society, 1994 , vol. 116, # 13 p. 6013 - 6014