反应条件
potassium hydroxide; hydrazine hydrate
1.) diethylene glycol, 150 deg C, 30 min., 2.) diethylene glycol, a) 150 deg C, 30 min., b) 210 deg C, 3 h; Yield given. Multistep reaction;
参考文献
Evans, Delme; Cracknell, Mark E.; Saunders, John C.; Smith, Christine E.; Williamson, W. R. Nigel; et al.
Journal of Medicinal Chemistry, 1987 , vol. 30, # 8 p. 1321 - 1327