反应条件
1: CuI; Cs2CO3; 1,3-bis(2,6-diisopropylphenyl)imidazolium chloride / Pd(OAc)2 / toluene / 2 h / 105 °C
2: 140 mg / CuI; 1,3-bis(2,6-diisopropylphenyl)imidazolium chloride; KOt-Bu / Pd(OAc)2 / toluene / 21 h / 105 °C
View Scheme
参考文献
Kaspar, Ludwig T.; Ackermann, Lutz
Tetrahedron, 2005 , vol. 61, # 48 p. 11311 - 11316