反应条件
1: 37 percent / methyl benzoylformate / acetonitrile; H2O / Ambient temperature
2: 1) 1-benzyl-1,4-dihydronicotinamide, 2) aq. HCl / 1) MeCN-H2O, room temp.
View Scheme
参考文献
Endo, Takeshi; Takada, Tadayoshi; Okawara, Makoto
Tetrahedron Letters, 1986 , vol. 27, # 5 p. 615 - 618