反应条件
1: 95 percent / 180 °C 2: 1.) N-bromosuccinimide, HF, pyridine, 2.) t-BuOK / 1.) ether, RT, 2 h, 2.) THF, from -30 deg C to -20 deg C, 2 h 3: 33 percent / 1 N aq. HCl / 19 h / 85 °C View Scheme
参考文献
Silverman; Bichler; Leon
Journal of the American Chemical Society, 1996 , vol. 118, # 6 p. 1241 - 1252