反应条件
1: 57.3 percent / POCl3, 2,4-dimethylpiperidine / 16 h / Heating
2: propan-2-ol / 1.) 2 h, 20 deg C, 2.) 30 min, 60 deg C
View Scheme
参考文献
Wollweber; Horstmann; Stoepel; Garthoff; Puls; Krause; Thomas
Arzneimittel-Forschung, 1981 , vol. 31, # 2 p. 279 - 288