1: With pyridine T=5 - 25°C; Neber Rearrangement; 2: With potassium tert-butylate in methanol T=10 - 25°C; Neber Rearrangement; 3: With hydrogenchloride in water T=80°C; 3 h;
参考文献
BIAL - PORTELA and Cª, S.A.; RUSSO, Domenico; WAHNON, Jorge Bruno Reis; MATON, William; ESZENYI, Tibor
Patent: WO2014/17938 A2, 2014 ;
Location in patent: Page/Page column 64; 65 ;