反应条件
1: With 1,1-dimethylethylmagnesium chloride; ethyl magnesium chloride in tetrahydrofuran
T=-78°C;
2: With N,N,N',N',N'',N''-hexamethylphosphoric triamide; PhSO2C(Li)HPh in tetrahydrofuran
T=-78 - 20°C;
参考文献
Satoh, Tsuyoshi; Sakamoto, Tatsuya; Watanabe, Masanori; Takano, Koji
Chemical and Pharmaceutical Bulletin, 2003 , vol. 51, # 8 p. 966 - 970