反应条件
1: triethylamine; ammonium chloride; 1-hydroxy-7-aza-benzotriazole; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride / N,N-dimethyl-formamide / 15 h / 0 - 20 °C
2: palladium on activated charcoal; hydrogen / methanol
View Scheme
参考文献
Teno, Naoki; Gohda, Keigo; Wanaka, Keiko; Tsuda, Yuko; Sueda, Takuya; Yamashita, Yukiko; Otsubo, Tadamune
Bioorganic and Medicinal Chemistry, 2014 , vol. 22, # 7 p. 2339 - 2352
