1: 92 percent / dioxane / 60 °C 2: 97 percent / 4-(dimethylamino)pyridine / methanol / 3 h / 60 °C View Scheme
参考文献
Venuti, Michael C.; Stephenson, Robert A.; Alvarez, Robert; Bruno, John J.; Strosberg, Arthur M.
Journal of Medicinal Chemistry, 1988 , vol. 31, # 11 p. 2136 - 2145
1: 96 percent / 150 °C 2: 75 percent / phosphorus oxychloride; N,N-diethylaniline / 4 h / Heating View Scheme
参考文献
Venuti, Michael C.; Stephenson, Robert A.; Alvarez, Robert; Bruno, John J.; Strosberg, Arthur M.
Journal of Medicinal Chemistry, 1988 , vol. 31, # 11 p. 2136 - 2145