1: triethylamine / dichloromethane / 20 °C
2: hydrogenchloride; water / dichloromethane / 20 °C
View Scheme
参考文献
Zulli, Allison L.; Aimone, Lisa D.; Mathiasen, Joanne R.; Gruner, John A.; Raddatz, Rita; Bacon, Edward R.; Hudkins, Robert L.
Bioorganic and Medicinal Chemistry Letters, 2012 , vol. 22, # 8 p. 2807 - 2810