N-（2-氨基苯甲酰基）甘氨酸合成路线 （共 18 条）
反应条件
hydrogenchloride; sodium nitrite in water Yield given;
参考文献
Susse; Johne
Helvetica Chimica Acta, 1985 , vol. 68, # 4 p. 892 - 899
反应条件
1: acetic acid / 2 h / 40 - 60 °C 2: 68 percent / KOH / ethanol; H2O / 2 h / Heating View Scheme
参考文献
Suesse, Manfred; Johne, Siegfried
Zeitschrift fuer Chemie (Stuttgart, Germany), 1985 , vol. 25, # 11 p. 403 - 404
反应条件
angiotensin I converting enzyme in water; dimethyl sulfoxide buffer (pH 8); Equilibrium constant;
参考文献
Sato; Nishikawa; Kanaoka
Chemical and Pharmaceutical Bulletin, 1989 , vol. 37, # 1 p. 145 - 147
反应条件
1: 6 h / Heating 2: 88 percent View Scheme
参考文献
Susse; Johne
Helvetica Chimica Acta, 1985 , vol. 68, # 4 p. 892 - 899
反应条件
Heating; Yield given;
参考文献
Susse; Johne
Helvetica Chimica Acta, 1985 , vol. 68, # 4 p. 892 - 899
反应条件
1: N-(2-aminobenzoyl)-glycine With pyridine; chloro-trimethyl-silane in dichloromethane T=25 - 30°C; 0.25 h; 2: p-pivaloyloxybenzenesulfonyl chloride in dichloromethane T=25 - 30°C; Further stages.;
参考文献
Bijukumar; Maloyesh; Sampat; Bhirud; Rajendra
Synthetic Communications, 2008 , vol. 38, # 11 p. 1718 - 1724
反应条件
sodium hydroxide in water
T=25 - 30°C; 0.5 h;
参考文献
Bijukumar; Maloyesh; Sampat; Bhirud; Rajendra
Synthetic Communications, 2008 , vol. 38, # 11 p. 1718 - 1724
反应条件
sodium hydroxide in water
T=70 - 80°C;
参考文献
DeRuiter, Jack; Swearingen, Blake E.; Wandrekar, Vinay; Mayfield, Charles A.
Journal of Medicinal Chemistry, 1989 , vol. 32, # 5 p. 1033 - 1038
反应条件
hydrogen; palladium on activated charcoal in ethanol; water
16 h;
参考文献
Locke, Darren; Bevans, Carville G.; Wang, Lai-Xi; Zhang, Ye; Harris, Andrew L.; Lee, Yuan C.
Carbohydrate Research, 2004 , vol. 339, # 2 p. 221 - 231
反应条件
1: oxalyl chloride; N,N-dimethylformamide / tetrahydrofuran / 2 h / 20 °C
2: 3.5 g / triethylamine / tetrahydrofuran / 5 h / 0 °C
3: H2 / Pd/C / ethanol; H2O / 16 h
View Scheme
参考文献
Locke, Darren; Bevans, Carville G.; Wang, Lai-Xi; Zhang, Ye; Harris, Andrew L.; Lee, Yuan C.
Carbohydrate Research, 2004 , vol. 339, # 2 p. 221 - 231
