反应条件
1: in N,N-dimethyl-formamide T=20°C; 2: With water in N,N-dimethyl-formamide T=20°C; 3: With sodium hydroxide in N,N-dimethyl-formamide T=20°C;
参考文献
AMGEN INC.; BROWN, Matthew; CHEN, Yi; CUSHING, Timothy D.; GONZALEZ LOPEZ DE TURISO, Felix; HE, Xiao; KOHN, Todd J.; LOHMAN, Julia Winslow; PATTAROPONG, Vatee; SEGANISH, Jennifer; SHIN, Youngsook; SIMARD, Jillian L.
Patent: WO2010/151737 A2, 2010 ;
Location in patent: Page/Page column 142 ;
WO 2010/151737 A2