反应条件
1: LiHMDS / THF 1) 1 h, -78 deg C 2) 2 h, -10 deg C 3) 1 h, -78 deg C 4) 16 h, r.t. 2: 82 percent / 0.5percent H2SO4 / acetic acid / 1 h / 95 - 100 °C View Scheme
参考文献
Ninomiya, Masayuki; Tanaka, Kaori; Tsuchida, Yuzo; Muto, Yoshinori; Koketsu, Mamoru; Watanabe, Kunitomo
Journal of Medicinal Chemistry, 2011 , vol. 54, # 5 p. 1529 - 1536