3-叔丁基-4-乙氧羰基咪唑合成路线 (共 1 条)
反应条件
1: lithium aluminium tetrahydride / tetrahydrofuran / 3 h / 20 °C 2: manganese(IV) oxide / acetone / 4 h / 20 °C 3: caesium carbonate / N,N-dimethyl-formamide / 5 h / 20 °C / Inert atmosphere 4: caesium carbonate View Scheme
参考文献
NEREUS PHARMACEUTICALS, INC.; YAMAZAKI, Yuri; HAYASHI, Yoshio
Patent: WO2011/84962 A1, 2011 ;