反应条件
1: 1.) NaH / 1.) DMF, RT, 30 min, 2.) DMF, RT, 1.5 h 2: t-BuOK / tetrahydrofuran / 16 h / Ambient temperature 3: 1.) n-Bu3SnH, palladium acetate, PPh3, 2.) Et4NCl*H2O / 1.) THF, 0 deg C, 1 h, 2.) acetonitrile, 80 deg C, 1 h View Scheme
参考文献
Grigg, Ronald; Sansano, Jose M.
Tetrahedron, 1996 , vol. 52, # 42 p. 13441 - 13454