1: With dichloro(1,1'-bis(diphenylphosphanyl)ferrocene)palladium(II) dichloromethane adduct in tetrahydrofuran T=50°C; 18 h; Inert atmosphere; 2: With water in tetrahydrofuran T=20°C;
参考文献
MERCK SHARP and DOHME CORP.; KUDUK, Scott, D.; CHANG, Ronald, K.; GRESHOCK, Thomas, J.
Patent: WO2012/47702 A1, 2012 ;
Location in patent: Page/Page column 39 ;
WO 2012/047702 A1