反应条件
1: 60 percent / 1M aq. NaOH / CHCl3; diethyl ether / 3 h / 0 °C
2: 42 percent / NaNO2, HCl / ethanol; H2O / 1.) 0 deg C, 30 min, 2.) 25 deg C, 1.5 h
View Scheme
参考文献
Sosnovsky; Rao
Journal of Pharmaceutical Sciences, 1991 , vol. 80, # 7 p. 693 - 699