反应条件
1: 1.) Et3N / 1.) DMF, -10 deg C, 2.) 20 deg C, 1 h
2: 92 percent / HCl / acetic acid / 1 h / 20 °C
View Scheme
参考文献
Sadovnikova, N. V.; Fedotov, V. P.; Shvachkin, Yu. P.; Shishkina, A. A.; Kolomeitseva, L. A.
Pharmaceutical Chemistry Journal, 1987 , vol. 21, # 12 p. 838 - 842
Khimiko-Farmatsevticheskii Zhurnal, 1987 , vol. 21, # 12 p. 1424 - 1427