2-氟-6-苯基吡啶-3-羧酸合成路线 (共 1 条)
反应条件
1: 2-fluoro-6-phenylpyridine With lithium diisopropyl amide in tetrahydrofuran
T=-78°C; 0.5 h;
2: carbon dioxide in tetrahydrofuran
0.166667 h;
参考文献
ELI LILLY AND COMPANY
Patent: WO2005/9941 A1, 2005 ;
Location in patent: Page 19 ;
WO 2005/009941 A1