反应条件
1: 2,4-dioxo-1,4-dihydro-2H-benzo[d][1,3]oxazine With sodium hydride in N,N-dimethyl-formamide
T=20°C; 1 h;
2: ethyl bromide in N,N-dimethyl-formamide
18 h;
参考文献
Clark, Rachel L.; Clements, Carol J.; Barrett, Michael P.; MacKay, Simon P.; Rathnam, Rajendra P.; Owusu-Dapaah, George; Spencer, John; Huggan, Judith K.
Bioorganic and Medicinal Chemistry, 2012 , vol. 20, # 20 p. 6019 - 6033