4-磺胺-5-甲氧基-6-氯嘧啶合成路线 (共 2 条)
反应条件
ammonia in water; butan-1-ol T=90°C; 2.5 h;
参考文献
MERCK SHARP and DOHME LIMITED
Patent: WO2005/47279 A1, 2005 ;
Location in patent: Page/Page column 33 ;
WO 2005/047279 A1
反应条件
sodium hydroxide in water T=65 - 70°C; 5 h; Heating / reflux; Product distribution / selectivity;
参考文献
DEGUSSA AG
Patent: WO2004/7466 A1, 2004 ;
Location in patent: Page/Page column 7-8 ;