甲基N2-[(苄氧基)羰基]天冬氨酰胺酰苯丙氨酸酯合成路线 （共 6 条）
反应条件
Sephadex G-50; triethylamine; bromelain in ethyl acetate
T=37°C; 7 h;
参考文献
Tai, Dar-Fu; Fu, Shu-Lin
Journal of the Chinese Chemical Society, 2003 , vol. 50, # 1 p. 179 - 183
反应条件
TEA in 1,4-dioxane
T=10°C; 0.5 h;
参考文献
Hartrodt; Neubert; Jakubke; Balaspiri; Telegdy
Pharmazie, 1982 , vol. 37, # 6 p. 403 - 407
参考文献
Pavo; Penke; Varga; et al.
Acta Chimica Hungarica, 1986 , vol. 122, # 3-4 p. 261 - 272
反应条件
triethylamine; 3-[(diethoxyphosphinyl)oxy]-1,2,3-benzotriazin-4(3H)-one
Ambient temperature;
参考文献
Fan, Chong-Xu; Hao, Xiao-Lin; Ye, Yun-Hua
Synthetic Communications, 1996 , vol. 26, # 7 p. 1455 - 1460
反应条件
1H-imidazole; triphenyl phosphite in N,N-dimethyl-formamide
参考文献
Yajima; Kiso; Kitagawa
Chemical and Pharmaceutical Bulletin, 1974 , vol. 22, # 5 p. 1079 - 1086
反应条件
(i) TsCl, HMPA, (ii) /BRN= 2212290/, Et3N; Multistep reaction;
参考文献
Gawne,G. et al.
Journal of the American Chemical Society, 1969 , vol. 91, # 20 p. 5669 - 5671
