1: 83.6 percent / K2CO3; NaI / acetone / 48 h / Heating
2: 86.5 percent / H2 / 10 percent Pd/C / ethanol / 20 °C / 760 Torr
3: KOH / ethanol / 20 °C
View Scheme
参考文献
Louis, Simon N.; Nero, Tracy L.; Iakovidis, Dimitri; Colagrande, Felicia M.; Jackman, Graham P.; Louis, William J.
European Journal of Medicinal Chemistry, 1999 , vol. 34, # 11 p. 919 - 937