3-胺基-5-溴苯并[D]异噁唑合成路线 (共 2 条)
反应条件
1: methanecarbohydroxamic acid With potassium tert-butylate in N,N-dimethyl-formamide T=30°C; 2: 3-cyano-4-fluoro-bromobenzene in N,N-dimethyl-formamide 3: With potassium tert-butylate in N,N-dimethyl-formamide
参考文献
WO2010/138488 A1, ;
Page/Page column 57-58 ;
WO 2010/138488 A1
反应条件
methanecarbohydroxamic acid; potassium tert-butylate in N,N-dimethyl-formamide T=20 - 50°C; 1.5 h;
参考文献
WO2006/122799 A1, ;
Page/Page column 60-61 ;