反应条件
1: N,N-dimethyl-formamide / Reflux 2: N-bromosuccinmide; 2,2'-azo-bisisobutyronitrile / 2 h / Reflux; Inert atmosphere View Scheme
参考文献
Zhang, Zhiyuan; Wallace, Michael B.; Feng, Jun; Stafford, Jeffrey A.; Skene, Robert J.; Shi, Lihong; Lee, Bumsup; Aertgeerts, Kathleen; Jennings, Andy; Xu, Rongda; Kassel, Daniel B.; Kaldor, Stephen W.; Navre, Marc; Webb, David R.; Gwaltney, Stephen L.
Journal of Medicinal Chemistry, 2011 , vol. 54, # 2 p. 510 - 524