1: 1-amino-4-methylthiobutane With triethylamine in tetrahydrofuran T=-10°C; Inert atmosphere; 2: carbon disulfide With dihydrogen peroxide in tetrahydrofuran T=-3 - 18°C;
参考文献
PHARMAGRA LABS, INC.; WELLS, Andrew; DAMIREDDI, Sahadeva Reddy; AKUE, Kpakpo Ambroise; NELSON, Jared K.; FRISBEE, Albert Roger; NEWSOME, Peter Wyatt
Patent: WO2013/179057 A1, 2013 ;
Location in patent: Paragraph 0098; 0099; 00100; 00101 ;