1,3,4,5-四氢-2H-1-苯并氮杂卓-2-酮合成路线 （共 62 条）
反应条件
titanium tetrachloride in tetrahydrofuran; benzene
参考文献
Collection of Czechoslovak Chemical Communications, , vol. 50, # 8 p. 1888 - 1898
反应条件
titanium tetrachloride in tetrahydrofuran; benzene
参考文献
Protiva; Sedivy; Holubek; et al.
Collection of Czechoslovak Chemical Communications, 1985 , vol. 50, # 8 p. 1888 - 1898
反应条件
AlCl3, aluminium chloride in carbon disulfide 3 h; Heating / reflux;
参考文献
WARNER-LAMBERT COMPANY LLC
Patent: WO2005/66165 A1, 2005 ;
Location in patent: Page/Page column 63 ;
参考文献
Pfizer Inc
Patent: US5350747 A1, 1994 ;
反应条件
1: 37.7 percent / sulfuryl chloride / benzene / 3 h / 20 °C 2: 88.1 percent / lithium aluminum hydride / tetrahydrofuran / 4 h / Heating View Scheme
参考文献
Ren, Hui; Zanger, Murray; McKee, James R.
Synthetic Communications, 2006 , vol. 36, # 3 p. 355 - 363
反应条件
lithium aluminium tetrahydride in tetrahydrofuran
参考文献
Robichaud, Albert J.; Lee, Taekyu; Deng, Wei; Mitchell, Ian S.; Chen, Wenting; McClung, Christopher D.; Calvello, Emilie J.; Zawrotny, David M.
Patent: US2004/209864 A1, 2004 ;
US 20040209864 A1
反应条件
BH3 in tetrahydrofuran
参考文献
Pfizer Inc.
Patent: US5736534 A1, 1998 ;
反应条件
1: 95 percent / TMSCl, NaI, I2, TMEDA / acetonitrile / -15 °C 2: 77 percent / NH3 / 100 °C View Scheme
参考文献
Armstrong, Joseph D. III; Eng, Kan K.; Keller, Jennifer L.; Purick, Robert M.; Hartner, Frederick W. Jr.; et al.
Tetrahedron Letters, 1994 , vol. 35, # 20 p. 3239 - 3242
反应条件
1: 68 percent / lithium aluminum hydride / tetrahydrofuran 2: 95 percent / HNO3; H2SO4 View Scheme
参考文献
Johnson, Paul D.; Aristoff, Paul A.; Zurenko, Gary E.; Schaadt, Ronda D.; Yagi, Betty H.; Ford, Charles W.; Hamel, Judith C.; Stapert, Douglas; Moerman, Judy K.
Bioorganic and Medicinal Chemistry Letters, 2003 , vol. 13, # 23 p. 4197 - 4200
反应条件
magnesium nitrate hexahydrate; potassium permanganate in water; tert-butyl alcohol 20 h; Ambient temperature;
参考文献
Chen; Gilman
Journal of Heterocyclic Chemistry, 1983 , vol. 20, # 3 p. 663 - 666
