反应条件
1: With 4-(N,N-dimethlyamino)pyridine; triethylamine in dichloromethane; N,N-dimethyl-formamide T=20°C; 24 h; 2: With trifluoroacetic acid in dichloromethane
参考文献
Parra, Andres; Martin-Fonseca, Samuel; Rivas, Francisco; Reyes-Zurita, Fernando J.; Medina-O'Donnell, Marta; Martinez, Antonio; Garcia-Granados, Andres; Lupianez, Jose A.; Albericio, Fernando
European Journal of Medicinal Chemistry, 2014 , vol. 74, p. 278 - 301