1: 68 percent / 2 h / 100 °C
2: 1) aqueous NH3; 2) AcOH / 1) Et2O, 2 h; 2) Et2O, 16 h
View Scheme
参考文献
Katritzky, Alan R.; Marson, Charles M.
Journal of the Chemical Society, Perkin Transactions 2: Physical Organic Chemistry (1972-1999), 1983 , # 9 p. 1455 - 1462
1: 65 percent / 5 h / 100 °C
2: 1) aqueous NH3; 2) AcOH / 1) Et2O, 2 h; 2) Et2O, 16 h
View Scheme
参考文献
Katritzky, Alan R.; Marson, Charles M.
Journal of the Chemical Society, Perkin Transactions 2: Physical Organic Chemistry (1972-1999), 1983 , # 9 p. 1455 - 1462