反应条件
trimethylsilyl bromide; diethyl cyanophosphonate; triethylamine
1) CH2Cl2, 18 h, room temperature; 2) DMF, 3 h, RT; 3) DMF, 12 d, RT; Yield given. Multistep reaction;
参考文献
Rosowsky; Forsch; Moran; Kohler; Freisheim
Journal of Medicinal Chemistry, 1988 , vol. 31, # 7 p. 1326 - 1331