6-氟-2-甲基-3-(4-甲基磺酰基-苄基)-1H-茚合成路线 (共 2 条)
反应条件
1: 70 percent / m-CPBA / CH2Cl2 / 1 h / 0 °C 2: Triton B / methanol / 12 h / 50 °C View Scheme
参考文献
Maguire; Papot; Ford; Touhey; O'Connor; Clynes
Synlett, 2001 , # 1 p. 41 - 44
反应条件
sodium hydroxide; sulfuric acid; iodine; magnesium in water; toluene
参考文献
FGN, INC.; THE UNIVERSITY OF ARIZONA
Patent: EP485172 A2, 1992 ;