1-CBZ-4-甲氨基哌啶合成路线 （共 3 条）
反应条件
1: With sodium tris(acetoxy)borohydride; acetic acid in 1,2-dichloro-ethane T=20°C; 2: With sodium hydrogencarbonate in water; 1,2-dichloro-ethane
参考文献
WO2009/76387 A1, ;
Page/Page column 40 ;
WO 2009/076387 A1
反应条件
1: in 1,4-dioxane; ethanol T=20°C; 0.25 h; 2: With sodium tris(acetoxy)borohydride in 1,4-dioxane; ethanol T=20°C; 15 h;
参考文献
WO2005/30209 A1, ;
Page/Page column 58 ;
WO 2005/030209 A1
反应条件
triethylamine in dichloromethane
T=20°C;
参考文献
GLAXO GROUP LIMITED
Patent: WO2009/76387 A1, 2009 ;
Location in patent: Page/Page column 40-41 ;
WO 2009/076387 A1
