反应条件
1: 1.) NaH / 1.) DMSO, 1 h, 2.) DMSO, RT, overnight
2: 1.) borane-THF, 2.) 12 N HCl / 1.) THF, reflux, 1 h, 2.) THF, reflux, 1 h
View Scheme
参考文献
Glamkowski, Edward J.; Fortunato, James M.; Spaulding, Theodore C.; Wilker, Jeffrey C.; Ellis, Daniel B.
Journal of Medicinal Chemistry, 1985 , vol. 28, # 1 p. 66 - 73