4-(4-氟苯基磺酰基)吗啉合成路线 (共 3 条)
参考文献
Wyeth
Patent: US2007/244140 A1, 2007 ;
Location in patent: Page/Page column 12 ;
反应条件
copper(ll) bromide in dimethyl sulfoxide T=100°C; 24 h; Inert atmosphere; chemoselective reaction;
参考文献
Tang, Xiaodong; Huang, Liangbin; Qi, Chaorong; Wu, Xia; Wu, Wanqing; Jiang, Huanfeng
Chemical Communications, 2013 , vol. 49, # 54 p. 6102 - 6104
反应条件
hydrazine in 1-methyl-pyrrolidin-2-one
T=100°C; 1 h;
参考文献
Schoenafinger, Karl; Petry, Stefan; Mueller, Guenter; Bauer, Armin; Heuer, Hubert Otto
Patent: US2003/236288 A1, 2003 ;
Location in patent: Page 18 ;
US 20030236288 A1