反应条件
1: sulfuric acid
2: lithium aluminium tetrahydride / tetrahydrofuran
3: 1H-imidazole / N,N-dimethyl-formamide
4: 1H-imidazole; iodine; triphenylphosphine / toluene
5: n-butyllithium; N,N,N',N',N'',N''-hexamethylphosphoric triamide / tetrahydrofuran
6: hydrogen; palladium on activated charcoal / ethyl acetate
7: pyridinium chlorochromate / dichloromethane
8: sodium hexamethyldisilazane / tetrahydrofuran
9: tetrabutyl ammonium fluoride / tetrahydrofuran
10: hydrogen; palladium 10 on activated carbon / ethyl acetate
View Scheme
参考文献
Zhang, Hong-Yan; Yamakawa, Yu-Ichiro; Matsuya, Yuji; Toyooka, Naoki; Tohda, Chihiro; Awale, Suresh; Li, Feng; Kadota, Shigetoshi; Tezuka, Yasuhiro
Bioorganic and Medicinal Chemistry Letters, 2014 , vol. 24, # 2 p. 604 - 608