2-溴-5-氟-3-甲基吡啶合成路线 (共 1 条)
反应条件
1.1: triethylamine / dichloro(1,1'-bis(diphenylphosphanyl)ferrocene)palladium(II) dichloromethane adduct / 20 h / 110 °C / 75007.5 Torr 2.1: water; lithium hydroxide hydrate / methanol / 16 h / 22 °C 2.2: pH 1 View Scheme
参考文献
Banner, David; Guba, Wolfgang; Hilpert, Hans; Humm, Roland; Mauser, Harald; Mayweg, Alexander V.; Narquizian, Robert; Power, Eoin; Rogers-Evans, Mark; Rombach, Didier; Woltering, Thomas; Wostl, Wolfgang
Patent: US2011/312937 A1, 2011 ;