反应条件
1: n-butyllithium; N,N,N',N,-tetramethylethylenediamine
2: hydrazine
3: 130 °C
4: iodine; potassium hydroxide / N,N-dimethyl-formamide / 2.5 h / 0 - 20 °C
View Scheme
参考文献
Herdemann, Matthias; Weber, Alexander; Jonveaux, Jerome; Schwoebel, Frank; Stoeck, Michael; Heit, Isabelle
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 6 p. 1852 - 1856
