(2S,5r)-1-(4-氟苄基)-2,5-二甲基哌嗪合成路线 (共 1 条)
反应条件
tetrabutylammomium bromide; sodium hydroxide in cyclohexane; water
T=35 - 45°C; 6 h; Inert atmosphere;
参考文献
Belecki, Katherine; Berliner, Martin; Bibart, Richard Todd; Meltz, Cliff; Ng, Karl; Phillips, James; Ripin, David H. Brown; Vetelino, Michael
Organic Process Research and Development, 2007 , vol. 11, # 4 p. 754 - 761