1.1: palladium (II) trifluoroacetate; silver trifluoromethanesulfonate / tetrahydrofuran; water / 24 h / 20 °C
1.2: 1 h / 20 °C
2.1: sodium tetrahydroborate / methanol / 1 h / 20 °C
View Scheme
参考文献
Ortega, Andrea; Rincon, Angela; Jimenez-Aliaga, Karim L.; Bermejo-Bescos, Paloma; Martin-Aragon, Sagrario; Molina, Maria Teresa; Csaky, Aurelio G.
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 8 p. 2183 - 2187