反应条件
1: 2,2,2-trifluoroethanol With sodium hydride in tetrahydrofuran T=20°C; 0.5 h; 2: (4-methoxyphenyl)phosphothioic dichloride in tetrahydrofuran T=20°C; Further stages.;
参考文献
Sawa, Masaaki; Tsukamoto, Takako; Kiyoi, Takao; Kurokawa, Kiriko; Nakajima, Fumio; Nakada, Yuichiro; Yokota, Koichi; Inoue, Yoshimasa; Kondo, Hirosato; Yoshino, Kohichiro
Journal of Medicinal Chemistry, 2002 , vol. 45, # 4 p. 930 - 936