反应条件
1: With bromine in tetrachloromethane; diethyl ether T=-10 - 20°C; 12.16 h; 2: With lithium carbonate; lithium bromide in N,N-dimethyl-formamide 3 h; Heating / reflux; 3: With hydrogenchloride in water T=0°C; pH=1;
参考文献
Kawakita, Youichi; Banno, Hiroshi; Ohashi, Tomohiro; Tamura, Toshiya; Yusa, Tadashi; Nakayama, Akiko; Miki, Hiroshi; Iwata, Hidehisa; Kamiguchi, Hidenori; Tanaka, Toshimasa; Habuka, Noriyuki; Sogabe, Satoshi; Ohta, Yoshikazu; Ishikawa, Tomoyasu
Journal of Medicinal Chemistry, 2012 , vol. 55, # 8 p. 3975 - 3991