3-氧代-3-苯基丙酰胺合成路线 (共 38 条)
反应条件
1: 3-methylthioaniline hydrochloride / toluene / Heating
2: diphenyl ether / 1 h / 240 °C
View Scheme
参考文献
Llinas-Brunet, Montse; Bailey, Murray D.; Ghiro, Elise; Gorys, Vida; Halmos, Ted; Poirier, Martin; Rancourt, Jean; Goudreau, Nathalie
Journal of Medicinal Chemistry, 2004 , vol. 47, # 26 p. 6584 - 6594
反应条件
1: m-trifluoromethylaniline hydrochloride / toluene / Heating
2: diphenyl ether / 1 h / 240 °C
View Scheme
参考文献
Llinas-Brunet, Montse; Bailey, Murray D.; Ghiro, Elise; Gorys, Vida; Halmos, Ted; Poirier, Martin; Rancourt, Jean; Goudreau, Nathalie
Journal of Medicinal Chemistry, 2004 , vol. 47, # 26 p. 6584 - 6594
反应条件
1: m-trifluoromethoxyaniline hydrochloride / toluene / Heating
2: diphenyl ether / 1 h / 240 °C
View Scheme
参考文献
Llinas-Brunet, Montse; Bailey, Murray D.; Ghiro, Elise; Gorys, Vida; Halmos, Ted; Poirier, Martin; Rancourt, Jean; Goudreau, Nathalie
Journal of Medicinal Chemistry, 2004 , vol. 47, # 26 p. 6584 - 6594
反应条件
1: m-acetamide aniline hydrochloride / toluene / Heating
2: diphenyl ether / 1 h / 240 °C
View Scheme
参考文献
Llinas-Brunet, Montse; Bailey, Murray D.; Ghiro, Elise; Gorys, Vida; Halmos, Ted; Poirier, Martin; Rancourt, Jean; Goudreau, Nathalie
Journal of Medicinal Chemistry, 2004 , vol. 47, # 26 p. 6584 - 6594
反应条件
1: m-bromoaniline hydrochloride / toluene / Heating
2: diphenyl ether / 1 h / 240 °C
View Scheme
参考文献
Llinas-Brunet, Montse; Bailey, Murray D.; Ghiro, Elise; Gorys, Vida; Halmos, Ted; Poirier, Martin; Rancourt, Jean; Goudreau, Nathalie
Journal of Medicinal Chemistry, 2004 , vol. 47, # 26 p. 6584 - 6594
参考文献
Obregia
Justus Liebigs Annalen der Chemie, 1891 , vol. 266, p. 329
反应条件
sodium hydrogencarbonate; pyruvic aldehyde in methanol; water
T=20°C; 22.5 h; Inert atmosphere;
参考文献
Kuramochi, Kouji; Sunoki, Takashi; Tsubaki, Kazunori; Mizushina, Yoshiyuki; Sakaguchi, Kengo; Sugawara, Fumio; Ikekita, Masahiko; Kobayashi, Susumu
Bioorganic and Medicinal Chemistry, 2011 , vol. 19, # 14 p. 4162 - 4172
参考文献
Obregia
Justus Liebigs Annalen der Chemie, 1891 , vol. 266, p. 329