1: With borane-THF in tetrahydrofuran 4 h; 2: With hydrogenchloride in tetrahydrofuran; water
参考文献
Pauly, Gary T.; Loktionova, Natalia A.; Fang, Qingming; Vankayala, Sai Lakshmana; Guida, Wayne C.; Pegg, Anthony E.
Journal of Medicinal Chemistry, 2008 , vol. 51, # 22 p. 7144 - 7153