反应条件
1: (COCl)2 / CH2Cl2 / 25 °C 2: 1,2-dichloro-ethane / 80 °C 3: 1.) KHMDS, 2.) TFA / tetrahydrofuran / 25 °C View Scheme
参考文献
Kulagowski; Baker; Curtis; Leeson; Mawer; Moseley; Ridgill; Rowley; Stansfield; Foster; Grimwood; Hill; Kemp; Marshall; Saywell; Tricklebank
Journal of Medicinal Chemistry, 1994 , vol. 37, # 10 p. 1402 - 1405