反应条件
1: 1,4-diaza-bicyclo[2.2.2]octane / ethanol / 20 °C / |Reflux 2: caesium carbonate / N,N-dimethyl-formamide / 7 h / 20 - 60 °C / |Inert atmosphere View Scheme
参考文献
Wang, Ning-Yu; Zuo, Wei-Qiong; Xu, Ying; Gao, Chao; Zeng, Xiu-Xiu; Zhang, Li-Dan; You, Xin-Yu; Peng, Cui-Ting; Shen, Yang; Yang, Sheng-Yong; Wei, Yu-Quan; Yu, Luo-Ting
Bioorganic and Medicinal Chemistry Letters, 2014 , vol. 24, # 6 p. 1581 - 1588