3-(4-羟基苯基)-2-[[2-(苯基甲氧羰基氨基)乙酰基]氨基]丙酸乙酯合成路线 （共 17 条）
反应条件
1,1'-carbonyldiimidazole
参考文献
Anderson et al.
Journal of the American Chemical Society, 1952 , vol. 74, p. 5304
Journal of the American Chemical Society, 1951 , vol. 73, p. 501
反应条件
1: 80 percent / HCl 2: 86 percent / DCC, HOBt / dimethylformamide / 24 h / 0 - 20 °C 3: 1) H2O2, acetone - H2O, 25 degC, 2 min, pH 9, 2) NaHSO3 View Scheme
参考文献
Roberts, David C.; Suda, Kohji; Samanen, James; Kemp, D. S.
Tetrahedron Letters, 1980 , vol. 21, p. 3435 - 3438
反应条件
1: 86 percent / DCC, HOBt / dimethylformamide / 24 h / 0 - 20 °C 2: 1) H2O2, acetone - H2O, 25 degC, 2 min, pH 9, 2) NaHSO3 View Scheme
参考文献
Losse,G. et al.
Justus Liebigs Annalen der Chemie, 1964 , vol. 677, p. 185 - 190
反应条件
1: 86 percent / DCC, HOBt / dimethylformamide / 24 h / 0 - 20 °C 2: 1) H2O2, acetone - H2O, 25 degC, 2 min, pH 9, 2) NaHSO3 View Scheme
参考文献
Roberts, David C.; Suda, Kohji; Samanen, James; Kemp, D. S.
Tetrahedron Letters, 1980 , vol. 21, p. 3435 - 3438
反应条件
triethylamine in chloroform
参考文献
Badiello,R. et al.
Gazzetta Chimica Italiana, 1964 , vol. 94, p. 322 - 327
反应条件
triethylamine in acetonitrile
参考文献
Losse,G. et al.
Justus Liebigs Annalen der Chemie, 1964 , vol. 677, p. 185 - 190
参考文献
Bergmann; Fruton
Journal of Biological Chemistry, 1937 , vol. 118, p. 405,414
反应条件
Ambient temperature;
参考文献
Chung-hsi, Li; Yuen-hwa, Yieh; Yao, Lin; Yong-jun, Lu; Ai-hsueh, Chi; Chi-yi, Hsing
Tetrahedron Letters, 1981 , vol. 22, # 36 p. 3467 - 3470
参考文献
Handford; Jones; Young; Johnson
Journal of the Chemical Society. Perkin transactions 1, 1965 , p. 6814 - 6827
反应条件
(i) PCl3, Py, (ii) /BRN= 4725904/; Multistep reaction;
参考文献
Yamazaki,N.; Higashi,F.
Bulletin of the Chemical Society of Japan, 1973 , vol. 46, # 12 p. 3821 - 3824
