反应条件
1: N,N-bis(trimethylsilyl)-2-aminothiazole With n-butyllithium in tetrahydrofuran T=-78°C; 0.5 h; 2: N,N-dimethyl-formamide in tetrahydrofuran T=-78 - -5°C; 0.5 h; 3: With hydrogenchloride in tetrahydrofuran Further stages.;
参考文献
Chen, Yuhpyng L.; Cherry, Kevin; Corman, Michael L.; Ebbinghaus, Charles F.; Gamlath, Chandra B.; Liston, Dane; Martin, Barbara-Anne; Oborski, Christine E.; Sahagan, Barbara G.
Bioorganic and Medicinal Chemistry Letters, 2007 , vol. 17, # 20 p. 5518 - 5522
