反应条件
thionyl chloride in N,N,N',N',N'',N''-hexamethylphosphoric triamide; acetonitrile
T=-5 - 0°C; 0.5 h;
参考文献
Takada, Susumu; Sasatani, Takashi; Chomei, Nobuo; Adachi, Makoto; Fujishita, Toshio; Eigyo, Masami; Murata, Shunji; Kawasaki, Kazuo; Matsushita, Akira
Journal of Medicinal Chemistry, 1996 , vol. 39, # 14 p. 2844 - 2851