反应条件
1: 1.) BuLi, 2.) iodine / 1) THF, hexane, 1.5 h, 0 deg C; 2) THF, hexane, 40 min, 0 deg C, room temperature, 2 h 2: Cu (powder) / Heating View Scheme
参考文献
Banzatti; Carfagna; Commisso; Heidempergher; Pegrassi; Melloni
Journal of Medicinal Chemistry, 1988 , vol. 31, # 7 p. 1466 - 1471